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CORRELATING DIFFERENTIAL ENDOGENOUS METABOLITE PROFILES WITH THE PHARMACOKINETICS OF GEFITINIB AND ITS ASSOCIATED DRUG METABOLITES USING AN ION MOBILITY BASED APPROACH

 

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Application Note LipidQuan™: A Robust LC-MS/MS Methodology for Rapidly Profiling the Lipidome of Liver Tissue Following Metabolism of the Drug Gefitinib Nyasha Munjoma, I.D. Wilson, Lee A. Gethings, Robert S. Plumb Waters Corporation For research use only. Not for use…
Key words
gefitinib, gefitinibmetabolism, metabolismdrug, druglipidomix, lipidomixtyrosine, tyrosineepidermal, epidermalliver, liverkinase, kinasenegative, negativegefitnib, gefitnibmultivatiate, multivatiategrowth, growthcommencement, commencementtkis, tkisxevo
LIPIDOMIC AND DESI IMAGING STUDY OF MOUSE LIVER DOSED WITH A TYROSINE KINASE INHIBITING DRUG Nyasha Munjoma 1 , Giorgis Isaac 2 , Mark Towers 1 , Emmanuelle Claude 1 , Ian D Wilson 3 , Lee A. Gethings 1…
Key words
desi, desiimaging, imaginguntargeted, untargetedgefitinib, gefitiniblipidomics, lipidomicstissue, tissueccs, ccslipid, lipidkinase, kinasepremier, premiergefitnib, gefitnibstatistical, statisticaltreated, treatedomics, omicstyrosine
Application Note Rapid Identification of Major Metabolites of Gefitinib Using Ion Mobility Enabled MS (HDMSE) with the SYNAPT XS Robert S. Plumb, Lauren Mullin, Adam King, Ian D. Wilson Waters Corporation, Computational and Systems Medicine, Imperial College Abstract This application…
Key words
synapt, synaptgefitinib, gefitinibunifi, unifienabled, enabledmobility, mobilityhdmse, hdmsemetabolite, metaboliteidentification, identificationresolution, resolutionccs, ccsmetabolites, metabolitesims, imsspectrometer, spectrometerquinazoline, quinazolinerelated
[ APPLICATION NOTE ] Analysis of Rat Urine Using Rapid Microbore Metabolic Profiling (RAMMP) HILIC Chromatography with Ion Mobility-MS Adam King, 1 Lauren Mullin, 2 Paul Rainville, 2 Robert Plumb, 2 Ian Wilson3 1 Waters Corporation, Wilmslow, UK 2 Waters…
Key words
rammp, rammphilic, hilicprofiling, profilingmetabolic, metabolicmicrobore, microboremobility, mobilityrat, ratrapid, rapidincreased, increasedurine, urineccs, ccsims, imschromatography, chromatographyopls, oplsion
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