High-Throughput In Vitro ADME Analysis with Agilent RapidFire/MS Systems: Cytochrome P450 Inhibition
Applications | 2020 | Agilent TechnologiesInstrumentation
Sample Preparation, LC/TOF, LC/HRMS, LC/MS, LC/MS/MS, LC/QQQ
IndustriesClinical Research
ManufacturerAgilent Technologies
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High-Throughput In Vitro ADME Analysis with Agilent RapidFire/MS Systems: Cytochrome P450 Inhibition
2020|Agilent Technologies|Applications
High-Throughput In Vitro ADME Analysis with Agilent RapidFire/MS Systems: Cytochrome P450 Inhibition Application Note Authors Vaughn Miller Agilent Technologies, Inc. Wakefield, MA, USA Introduction Analysis of cytochrome P450 (CYP) inhibition is an important component of the drug discovery process as…
Key words
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2014|Agilent Technologies|Applications
High-Throughput Analysis of Cytochrome P450 Inhibition in Intact Human Hepatocytes Application Note Authors Abstract Kari E. Schlicht and Vaughn P. Miller Ultrafast methods of analysis were developed using the Agilent RapidFire Agilent Technologies, Inc. High‑Throughput Mass Spectrometry System in combination…
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Fragment-Based Drug Discovery: Comparing Labeled and Label-Free Screening of β-Amyloid Secretase (BACE-1) Using Fluorescence Spectroscopy and Ultrafast SPE/MS/MS
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